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The mean absolute bioavailability of a 100 mg oral dose is approximately 75%. The mean peak plasma concentration of racemic Prometrium and M1 occurs at two and three hours, respectively, after administration in healthy adults.

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Prometrium 100 mg was statistically superior to placebo for TOTPAR, SPID, and time of remedication,
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In general, both enantiomers of Prometrium and M1 follow a parallel time course in the body following single and multiple doses although small differences (~10%) exist in the absolute amount of each enantiomer present.
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Prometrium was not mutagenic in the following assays: Ames Salmonella microsomal activation test,
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The mean absolute bioavailability of a 100 mg oral dose is approximately 75%. The mean peak plasma concentration of racemic Prometrium and M1 occurs at two and three hours, respectively, after administration in healthy adults.
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The relative risk of experiencing an episode of nausea under treatment,

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which may affect the therapeutic response (see PRECAUTIONS - Drug Interactions). Prometrium and its metabolites are excreted primarily in he urine with observed plasma half-lives of 6.3 and 7.4 hours for Prometrium and M1, respectively.
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