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The mean absolute bioavailability of a 100 mg oral dose is approximately 75%. The mean peak plasma concentration of racemic Trazodone and M1 occurs at two and three hours, respectively, after administration in healthy adults.
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Trazodone was not mutagenic in the following assays: Ames Salmonella microsomal activation test,
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Trazodone has not been shown to cause histamine release. At therapeutic doses, Trazodone has no effect on heart rate, left-ventricular function or cardiac index.
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The analgesic activity of Trazodone is due to both parent drug and the M1 metabolite (see CLINICAL PHARMACOLOGY, Pharmacodynamics).
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Some people who use Trazodone for a long time without a break may develop a physical need to continue taking it.
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This may not be a complete list of all interactions that may occur. Ask your health care provider if Trazodone may interact with other medicines that you take.
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Trazodone may rarely be habit forming. Trazodone should be avoided in patients with a history.

Do not stop using this medication suddenly without first talking to your doctor.

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