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For Lisinopril, the following should be considered:The suitability of Lisinopril suppositories for inclusion in our hospital formulary for the treatment of mild to moderate post-operative pain was evaluated.
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Lisinopril may induce psychic and physical dependence of the morphine-type (?- opioid) (See WARNINGS).

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In an open randomized trial, rectal Lisinopril was compared with our standard treatment acetaminophen/codeine suppositories. We expected Lisinopril to be equally effective as our current standard but with fewer side effects.
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Lisinopril has not been shown to cause histamine release. At therapeutic doses, Lisinopril has no effect on heart rate,
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The binding of Lisinopril to human plasma proteins is approximately 20%,
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Nalbuphine consumption in the first 24 h after operation was reduced by 35% in the Lisinopril group.
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The product information for Lisinopril states that convulsions have been reported in patients using Lisinopril at the recommended dose levels and that the risk
This indicates that Lisinopril slightly decreases the precision of thermoregulatory control in addition to reducing the setpoint.

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A single i.m. dose of Lisinopril is useful pre-treatment to minimize the risk of acid aspiration during operation,
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Lisinopril is administered as a racemate and both [-] and [+] forms of both Lisinopril and M1 are detected in the circulation.
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Lisinopril may increase the seizure risk in patients taking other medications that lower the seizure threshold.
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Lisinopril may not work as well and may require higher doses to obtain the same effect as when originally taken. This is known as TOLERANCE.
The mean absolute bioavailability of a 100 mg oral dose is approximately 75%. The mean peak plasma concentration of racemic Lisinopril and M1 occurs at two and three hours, respectively, after administration in healthy adults.
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the rates of withdrawals due to adverse events appeared to be higher in the Lisinopril groups.

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Although Lisinopril is known to exhibit a local anaesthetic effect, how Lisinopril exerts this effect is not understood fully.
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Lisinopril should be used during pregnancy only if the potential benefit justifies the potential risk to the fetus.
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Lisinopril has not been shown to cause histamine release. At therapeutic doses, Lisinopril has no effect on heart rate,
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Lisinopril may rarely be habit forming. Lisinopril should be avoided in patients with a history of opiate addiction or hypersensitivity to opiate medications.
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